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Automating drug discovery | Nature Reviews Drug Discovery
Automating drug discovery | Nature Reviews Drug Discovery

Biophysics in drug discovery: impact, challenges and opportunities | Nature  Reviews Drug Discovery
Biophysics in drug discovery: impact, challenges and opportunities | Nature Reviews Drug Discovery

Investigating antimalarial drug interactions of emetine dihydrochloride  hydrate using CalcuSyn-based interactivity calculations
Investigating antimalarial drug interactions of emetine dihydrochloride hydrate using CalcuSyn-based interactivity calculations

An in vitro toolbox to accelerate anti-malarial drug discovery and  development | Malaria Journal | Full Text
An in vitro toolbox to accelerate anti-malarial drug discovery and development | Malaria Journal | Full Text

Screening-based approach to discover effective platinum-based  chemotherapies for cancers with poor prognosis
Screening-based approach to discover effective platinum-based chemotherapies for cancers with poor prognosis

Covalent fragment libraries in drug discovery - ScienceDirect
Covalent fragment libraries in drug discovery - ScienceDirect

Drug development - Wikipedia
Drug development - Wikipedia

Computational design of substrate selective inhibition
Computational design of substrate selective inhibition

Mechanistic enzymology in drug discovery: a fresh perspective | Nature  Reviews Drug Discovery
Mechanistic enzymology in drug discovery: a fresh perspective | Nature Reviews Drug Discovery

Recent advances in combinatorial drug screening and synergy scoring -  ScienceDirect
Recent advances in combinatorial drug screening and synergy scoring - ScienceDirect

Effects of target binding kinetics on in vivo drug efficacy: koff, kon and  rebinding - Vauquelin - 2016 - British Journal of Pharmacology - Wiley  Online Library
Effects of target binding kinetics on in vivo drug efficacy: koff, kon and rebinding - Vauquelin - 2016 - British Journal of Pharmacology - Wiley Online Library

The drug–target residence time model: a 10-year retrospective | Nature  Reviews Drug Discovery
The drug–target residence time model: a 10-year retrospective | Nature Reviews Drug Discovery

Biased Receptor Signaling in Drug Discovery | Pharmacological Reviews
Biased Receptor Signaling in Drug Discovery | Pharmacological Reviews

CISNE: An accurate description of dose-effect and synergism in combination  therapies | Scientific Reports
CISNE: An accurate description of dose-effect and synergism in combination therapies | Scientific Reports

The nature of ligand efficiency | SpringerLink
The nature of ligand efficiency | SpringerLink

DeepConv-DTI: Prediction of drug-target interactions via deep learning with  convolution on protein sequences
DeepConv-DTI: Prediction of drug-target interactions via deep learning with convolution on protein sequences

Automating drug discovery | Nature Reviews Drug Discovery
Automating drug discovery | Nature Reviews Drug Discovery

Macrocycles in new drug discovery | Future Medicinal Chemistry
Macrocycles in new drug discovery | Future Medicinal Chemistry

The implications of target saturation for the use of drug–target residence  time | Nature Reviews Drug Discovery
The implications of target saturation for the use of drug–target residence time | Nature Reviews Drug Discovery

Creating and screening natural product libraries - Natural Product Reports  (RSC Publishing) DOI:10.1039/C9NP00068B
Creating and screening natural product libraries - Natural Product Reports (RSC Publishing) DOI:10.1039/C9NP00068B

PDF) Theoretical Basis, Experimental Design, and Computerized Simulation of  Synergism and Antagonism in Drug Combination Studies
PDF) Theoretical Basis, Experimental Design, and Computerized Simulation of Synergism and Antagonism in Drug Combination Studies

A Comprehensive Biophysical Analysis of the Effect of DNA Binding Drugs on  Protamine-induced DNA Condensation | Scientific Reports
A Comprehensive Biophysical Analysis of the Effect of DNA Binding Drugs on Protamine-induced DNA Condensation | Scientific Reports

Direct small-molecule inhibitors of KRAS: from structural insights to  mechanism-based design | Nature Reviews Drug Discovery
Direct small-molecule inhibitors of KRAS: from structural insights to mechanism-based design | Nature Reviews Drug Discovery

Recent advances in combinatorial drug screening and synergy scoring -  ScienceDirect
Recent advances in combinatorial drug screening and synergy scoring - ScienceDirect

The drug–target residence time model: a 10-year retrospective | Nature  Reviews Drug Discovery
The drug–target residence time model: a 10-year retrospective | Nature Reviews Drug Discovery

Covalent fragment libraries in drug discovery - ScienceDirect
Covalent fragment libraries in drug discovery - ScienceDirect